WO2006044856A2 - Use of a2a adenosine receptor agonists - Google Patents
Use of a2a adenosine receptor agonists Download PDFInfo
- Publication number
- WO2006044856A2 WO2006044856A2 PCT/US2005/037368 US2005037368W WO2006044856A2 WO 2006044856 A2 WO2006044856 A2 WO 2006044856A2 US 2005037368 W US2005037368 W US 2005037368W WO 2006044856 A2 WO2006044856 A2 WO 2006044856A2
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- WO
- WIPO (PCT)
- Prior art keywords
- pharmaceutical composition
- regadenoson
- human
- single dose
- administered
- Prior art date
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/22—Echographic preparations; Ultrasound imaging preparations ; Optoacoustic imaging preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Physics & Mathematics (AREA)
- Acoustics & Sound (AREA)
- Radiology & Medical Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Saccharide Compounds (AREA)
Abstract
Description
Claims
Priority Applications (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05815368A EP1802317A2 (en) | 2004-10-20 | 2005-10-19 | Use of a2a adenosine receptor agonists |
CA002583185A CA2583185A1 (en) | 2004-10-20 | 2005-10-19 | Use of a2a adenosine receptor agonists |
MX2007004749A MX2007004749A (en) | 2004-10-20 | 2005-10-19 | Use of a2a adenosine receptor agonists. |
JP2007537961A JP2008517063A (en) | 2004-10-20 | 2005-10-19 | Use of A2A adenosine receptor agonist |
AU2005295437A AU2005295437B2 (en) | 2004-10-20 | 2005-10-19 | Use of A2A adenosine receptor agonists |
IL182645A IL182645A0 (en) | 2004-10-20 | 2007-04-18 | Use of a2a adenosine receptor agonists |
NO20072540A NO20072540L (en) | 2004-10-20 | 2007-05-18 | Use of A2A adenosine receptor agonist |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US62057704P | 2004-10-20 | 2004-10-20 | |
US60/620,577 | 2004-10-20 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2006044856A2 true WO2006044856A2 (en) | 2006-04-27 |
WO2006044856A3 WO2006044856A3 (en) | 2006-07-06 |
Family
ID=35953984
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2005/037368 WO2006044856A2 (en) | 2004-10-20 | 2005-10-19 | Use of a2a adenosine receptor agonists |
Country Status (13)
Country | Link |
---|---|
US (3) | US7655636B2 (en) |
EP (1) | EP1802317A2 (en) |
JP (1) | JP2008517063A (en) |
KR (1) | KR20070083714A (en) |
CN (1) | CN101076343A (en) |
AU (1) | AU2005295437B2 (en) |
CA (1) | CA2583185A1 (en) |
IL (1) | IL182645A0 (en) |
MX (1) | MX2007004749A (en) |
NO (1) | NO20072540L (en) |
RU (1) | RU2007114908A (en) |
WO (1) | WO2006044856A2 (en) |
ZA (1) | ZA200703229B (en) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2066232A1 (en) * | 2006-09-29 | 2009-06-10 | Cv Therapeutics, Inc. | Methods for myocardial imaging in patients having a history of pulmonary disease |
JP2010515081A (en) * | 2007-01-03 | 2010-05-06 | ギリアード・パロ・アルト・インコーポレイテッド | Myocardial perfusion imaging |
US8071566B2 (en) | 2000-02-23 | 2011-12-06 | Gilead Sciences, Inc. | Methods of coronary imaging |
RU2459626C2 (en) * | 2006-09-01 | 2012-08-27 | Гайлид Сайэнсиз, Инк. | Methods and compositions improving patient's tolerance of myocardial visualisation technique |
US8906878B2 (en) | 2002-07-29 | 2014-12-09 | Gilead Sciences, Inc. | Myocardial perfusion imaging methods and compositions |
USRE47301E1 (en) | 2006-02-03 | 2019-03-19 | Gilead Sciences, Inc. | Process for preparing an A2A-adenosine receptor agonist and its polymorphs |
USRE47351E1 (en) | 1999-06-22 | 2019-04-16 | Gilead Sciences, Inc. | 2-(N-pyrazolo)adenosines with application as adenosine A2A receptor agonists |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6403567B1 (en) | 1999-06-22 | 2002-06-11 | Cv Therapeutics, Inc. | N-pyrazole A2A adenosine receptor agonists |
US6214807B1 (en) * | 1999-06-22 | 2001-04-10 | Cv Therapeutics, Inc. | C-pyrazole 2A A receptor agonists |
CA2492855C (en) * | 2002-07-29 | 2012-09-18 | Cv Therapeutics, Inc. | Myocardial perfusion imaging using a2a receptor agonists |
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US8106029B2 (en) | 2012-01-31 |
US20060084625A1 (en) | 2006-04-20 |
IL182645A0 (en) | 2007-07-24 |
KR20070083714A (en) | 2007-08-24 |
JP2008517063A (en) | 2008-05-22 |
MX2007004749A (en) | 2007-06-18 |
US20100158797A1 (en) | 2010-06-24 |
CA2583185A1 (en) | 2006-04-27 |
WO2006044856A3 (en) | 2006-07-06 |
ZA200703229B (en) | 2009-07-29 |
US7655636B2 (en) | 2010-02-02 |
CN101076343A (en) | 2007-11-21 |
AU2005295437A1 (en) | 2006-04-27 |
NO20072540L (en) | 2007-05-18 |
EP1802317A2 (en) | 2007-07-04 |
US20120189538A1 (en) | 2012-07-26 |
RU2007114908A (en) | 2008-10-27 |
AU2005295437B2 (en) | 2011-05-19 |
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